参考文献/References:
1 Tua Z,Dencea C,Ponde D,et al.Carbon-11 labeled r2 receptor ligands for imaging breast cancer.Nucl Med Biol,2005,32(5):423-430.
2 Mading P,Zessin J,Plei U,et al.Synthesis of a 11C-labelled taxane derivative by[1-11C] acetylation.J Label Compd Radio-pharm,2006,49(4):357-365.
3 Zimme L,Fournet G,Joseph B,et al.Carbon-11 labelling of 8{{3-[4-(2-[11C] methoxyphenyl) piperazin-1-yl]-2-hydroxypropyl}oxy} thiochroman,a presynaptic 5-HT1A receptoragonist,and its in vivo evaluation in anaesthetised rat and in awake cat.Nucl Med Biol,2003,30(5):541-546.
4 Bolton R.Isotopic methylation.J Label Compd Radiopharm,2001,44(10):701-736.
5 Iwata R,Pascalic C,Bogni A,et al.A simple loop method for the automated preparation of[11C] raclopride from[11C] methyl triflate.Appl Radiat Isot,2001,55(1):17-22.
6 Langer O,Nagren K,Dolle F,et al.Precursor synthesis and radiolabelling of the dopamine D2 receptor ligand 11C-raclopride from 11C-methyl Triflate.J Label Compd Radiopharm,1999,42(12):1183-1193.
7 Matattese M,Soloviev D,Moresco RM,et al.Synthesis and vivo evaluation of 3-11C-methyl-(3-methyoxy-naphthalen-2-gl-(1-benzylpiperidin)-4-yl-acetate (SB-235753),as a putative dopamine D4receptor antagonist for PET.J Label Compd Radiopharm,2000,43(4):359.
8 Dolle F,Bramoulle Y,Hinnen F,et al.Efficient synthesis and formulation of (R)-(-)-[11C] Deprenyl,a selectiveradioligand for the quantification of MAO-B activity using PET.J Label Compd Radiopharm,2002,45(10):803-811.
9 Nagren K,Muller L,Halldon C,et al.Improved synthesis of some commonly used PET radioligands by the use of 11C-methyl triflate.Nucl Med Boil,1995,22(2):235-239.
10 Lundkvist C,Halldin C,Swahn CG,et al.Improved synthesis of the PET radioligands 11C-FLB457,11C-MDL100907 and 11C-CIT-FE by use of 11C-methyl Triflate.J Label Compd Radiopharm,1998,41(6):545-556.
11 Luurtsemal G,Windhorst AD,Martien PJ,et al.Fully automated high yield synthesis of (R)- and (S)-[11C]verapamil for measuring Pglycoprotein function with positron emission tom-ography.J Label Compd Radiopharm,2002,45(14):1199-1207.
12 Solbach C,Uebele M,Reisch G,et al.Efficient radiosynthesis of carbon-11 labelled uncharged thioflavin T derivatives using[11C] methyl triflate for β-amyloid imaging in Alzheimer’s disease with PET.Appl Radiat Isot,2005,62(4):591-595.
13 Klunk W,Wang Y,Huang G,et al.Uncharged thioflavin-T derivatives bind to amyloid-beta protein with high affinity and readily enter the brain.Life Sci,2001,69(13):1471-1484.
14 Mathis CA,Wang Y,Holt DP,et al.Synthesis and evaluation of 11C-labeled 6-substituted 2-arylbenzothiazoles as amyloid imaging agents.J Med Chem,2003,46(13):2740-2754.
15 Mathis CA,Bacskai BJ,Kajdasz ST,et al.A lipophilic ThioflavinT derivative for positron emission tomograph (PET) imaging of amy-loid in brain.Bioorg Med Chem Lett,2002,12(2):295-298.
16 Ishiwata K,Ishii S,Senda M.An alternative synthesis of[11C] raclopride for routine use.Ann Nucl Med,1999,13(3):195-197.
17 Schou M,Halldin C,S6vágo J,et al.Specific in vivo binding to the norepinephrine transporter demonstrated with the PET radioligand,(S,S)-[11C] MeNER.Nucl Med Biol,2003,30(7):707-714.
18 Elisinga PH,Van Warde A,Visser GM,et al.Synthesis and preliminary evaluation of (R,S)-1-[2-((carbamoyl-4-hydroxy) phenoxy)-ethylamino]-3-[4-(1-[11C]-methyl-4-trifluoromethyl-2-imidazolyl)phenoxy]-2-propanol(11C-CGP20712A) as a selective β1-adrenoceptor ligand for PET.Nucl Med Biol,1994,21(2):211-217.
19 Todde S,Moresco RM,Frostl W,et al.Synthesis and in vivo evaluation of[(11) C] CGP62349,a new GABA (B) receptor antagonist.Nucl Med Biol,2000,27(6):565-569.
20 Kuhnast B,Bodenstein C,Wester HJ.et al.Carbon-11 labelling of an N-sulfonylamino acidderivative:a potential tracer for MMP-2and MMP-9 imaging.J Label Compd Radiopharm,2003,46(6):539-553.
21 Wilson AA,Garcia A,Chestakova A,et al.A rapid one-step radiosynthesis of β-amyloid imaging radiotracer N-methyl-[11C] 2-(4’-methylaminophenyl)-6-hydroxy benzothiazlo([11C]-6-OH-BTA-1).J Label Compd Radiopharm,2004,47(10):679-682.
22 Wang YM,Mathis CA,Huang GF,et al.Synthesis and 11C-labelling of (E,E)-1-(3’,4’-dihydroxystyryl)-4-(3’-methoxy-4’-hydroxystyryl)benzene for PET imaging of amyloid deposits.J Label Compds Radiopharm,2002,45(8):647-664.
23 Bender D,Holschbach M,Stocklin G,et al.Synthesis of n.c.a carbon-11 labelled clozapine and its major metaboite clozapine-Noxide and comparison of their biodistribution in mice.Nucl Med Biol,1994,21(7):921-925.
24 Zhang JM,Tian JH,Wang WS,et al.A new technique for labeling of 11C-choline,a positron emiting tracer for tumor imaging.J Radioanal Nucl Med,2006,267(3):665-668.
25 Huang Y,Narendran R,Bae SA,et al.A PET imaging agent with fast kinetics:synthesis and in vivo evaluation of the serotonin transporter ligand[11C]2-(2-dimethylaminomethylphenylthio)-5-fluorophenylamine ([11C]AFA).Nucl Med Biol,2004,31(6):727-738.
26 Schweiger L,Craib S,Welch A,et al.Radiosynthesis of[Nmethyl-11C] methylene blue.J Label Compd Radiopharm,2003,46(13):1221-1228.
相似文献/References:
[1]李海峰,张晓军,李云钢,等.国产模块LOOP环改良法合成11C-蛋氨酸[J].国际放射医学核医学杂志,2016,40(2):106.[doi:10.3760/cma.j.issn.1673-4114.2016.02.004]
Li Haifeng,Zhang Xiaojun,Li Yungang,et al.Synthesis of 11C-methionine on home-made module by the improved LOOP method[J].International Journal of Radiation Medicine and Nuclear Medicine,2016,40(5):106.[doi:10.3760/cma.j.issn.1673-4114.2016.02.004]
[2]赵雷,杨雁,孙华.自动化固相萃取法合成11C-乙酸盐的影响因素[J].国际放射医学核医学杂志,2015,39(3):224.[doi:10.3760/cma.j.issn.1673-4114.2015.03.008]
Zhao Lei,Yang Yan,Sun Hua.Influential factors of solid-phase extraction method to automate the synthesis of 11C-acetate[J].International Journal of Radiation Medicine and Nuclear Medicine,2015,39(5):224.[doi:10.3760/cma.j.issn.1673-4114.2015.03.008]
[3]展凤麟,汪世存,潘博,等.11C-胆碱和18F-FDG PET/CT显像在脑胶质瘤诊断中的应用[J].国际放射医学核医学杂志,2013,37(4):193.[doi:10.3760/cma.j.issn.1673-4114.2013.04.001]
ZHAN Feng-lin,WANG Shi-cun,PAN Bo,et al.Application of 11C-choline and 18F-FDG PET/CT in diagnosing brain glioma[J].International Journal of Radiation Medicine and Nuclear Medicine,2013,37(5):193.[doi:10.3760/cma.j.issn.1673-4114.2013.04.001]
[4]孙爱君,任茜,刘健,等.11C-乙酸盐PET和PET/CT在肿瘤显像中的应用[J].国际放射医学核医学杂志,2013,37(4):243.[doi:10.3760/cma.j.issn.1673-4114.2013.04.013]
SUN Ai-jun,REN Qian,LIU Jian,et al.The application of 11C-acetate PET and PET-CT for tumors[J].International Journal of Radiation Medicine and Nuclear Medicine,2013,37(5):243.[doi:10.3760/cma.j.issn.1673-4114.2013.04.013]
[5]马文超,徐文贵.11C-乙酸盐在肿瘤PET或PET-CT中的应用[J].国际放射医学核医学杂志,2011,35(1):23.[doi:10.3760/cma.j.issn.1673-4114.2011.01.007]
MA Wen-chao,XU Wen-gui.The application of 11C-acetate PET or PET-CT for tumors[J].International Journal of Radiation Medicine and Nuclear Medicine,2011,35(5):23.[doi:10.3760/cma.j.issn.1673-4114.2011.01.007]
[6]李亚军,张慧娟.放射性核素标记胆碱与18F-FDG PET肿瘤显像的对比研究[J].国际放射医学核医学杂志,2010,34(6):348.[doi:10.3760/cma.j.issn.1673-4114,2010.06.007]
LI Ya-jun,ZHANG Hui-juan.Comparison choline with 18F-FDG PET in various tumors imaging[J].International Journal of Radiation Medicine and Nuclear Medicine,2010,34(5):348.[doi:10.3760/cma.j.issn.1673-4114,2010.06.007]